Vineet Pande

ScholarGPS® ID: 68158456506207

Affiliation

Janssen Pharmaceutica

Affiliation History

Field

Physical Sciences and Mathematics

Discipline

Chemistry

Top Specialties

Medicinal Chemistry | DNA | Androgen Receptor

Metrics Summary

Publication Count

Predicted Citations

736

Predicted h-index

Ranking

Publications and Citation History

Publications based on Top Specialties

Types of Publication

Publications
Books
Patents
NIH/NSF

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Gut-Restricted Selective Cyclooxygenase-2 (COX-2) Inhibitors for Chemoprevention of Colorectal Cancer (journal article) Zhang, Zhuming \| Ghosh, Avijit \| Connolly, Peter J. \| King, Peter \| Wilde, Thomas \| Wang, Jianyao \| Dong, Yawei \| Li, Xueliang \| Liao, Daohong \| Chen, Hao \| ... \| Evans, David C. Journal of Medicinal Chemistry, volume 64, issue 15, pages 11570-11596 (2021). 10.1021/acs.jmedchem.1c00890 Cited by (12) \| Cite \| Source
Spirocyclic Thiohydantoin Antagonists of F877L and Wild-Type Androgen Receptor for Castration-Resistant Prostate Cancer (journal article) Zhang, Zhuming \| Connolly, Peter J. \| Trabalón Escolar, Luis \| Rocaboy, Christian \| Pande, Vineet \| Meerpoel, Lieven \| Lim, Heng-Keang \| Branch, Jonathan R. \| Ondrus, Janine \| Hickson, Ian \| ... \| Bignan, Gilles ACS Medicinal Chemistry Letters, volume 12, issue 8, pages 1245-1252 (2021). 10.1021/acsmedchemlett.1c00032 Cited by (3) \| Cite \| Source
Preparation of Novel 4′-Spirocyclopropyl Nucleoside Analogues (journal article) Verhoeven, Jonas \| Kong, Hanchu \| Zhao, Yongbin \| Wang, Wenbin \| Pande, Vineet \| Brambilla, Marta \| Van Hecke, Kristof \| Meerpoel, Lieven \| Thuring, Jan Willem \| Verniest, Guido Synlett, volume 32, issue 09, pages 892-896 (2021). 10.1055/a-1386-7194 Cited by (6) \| Cite \| Source
Discovery of JNJ-63576253, a Next-Generation Androgen Receptor Antagonist Active Against Wild-Type and Clinically Relevant Ligand Binding Domain Mutations in Metastatic Castration-Resistant Prostate Cancer (journal article) Branch, Jonathan R. \| Bush, Tammy L. \| Pande, Vineet \| Connolly, Peter J. \| Zhang, Zhuming \| Hickson, Ian \| Ondrus, Janine \| Jaensch, Steffen \| Bischoff, James R. \| Habineza, Georges \| ... \| Bignan, Gilles Molecular Cancer Therapeutics, volume 20, issue 5, pages 763-774 (2021). 10.1158/1535-7163.MCT-20-0510 Cited by (3) \| Cite \| Source
Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC) (journal article) Zhang, Zhuming \| Connolly, Peter J. \| Lim, Heng Keang \| Pande, Vineet \| Meerpoel, Lieven \| Teleha, Christopher \| Branch, Jonathan R. \| Ondrus, Janine \| Hickson, Ian \| Bush, Tammy \| ... \| Bignan, Gilles Journal of Medicinal Chemistry, volume 64, issue 2, pages 909-924 (2021). 10.1021/acs.jmedchem.0c01563 Cited by (17) \| Cite \| Source
Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues (journal article) Verhoeven, Jonas \| Deraet, Xavier \| Pande, Vineet \| Sun, Weimei \| Alonso, Mercedes \| De Proft, Frank \| Meerpoel, Lieven \| Thuring, Jan Willem \| Verniest, Guido The Journal of Organic Chemistry, volume 85, issue 23, pages 14989-15005 (2020). 10.1021/acs.joc.0c01825 Cited by (2) \| Cite \| Source
A Chemical Probe for the Methyl Transferase PRMT5 with a Novel Binding Mode (journal article) Pande, Vineet \| Sun, Weimei \| Beke, Lijs \| Berthelot, Didier \| Brehmer, Dirk \| Brown, David \| Corbera, Jordi \| Irving, Steve \| Meerpoel, Lieven \| Nys, Thomas \| ... \| Thuring, Jan Willem ACS Medicinal Chemistry Letters, volume 11, issue 11, pages 2227-2231 (2020). 10.1021/acsmedchemlett.0c00355 Cited by (14) \| Cite \| Source
Azepane inhibitors of menin-MLL interaction (patent) Angibaud, Patrick René \| Pande, Vineet \| Herkert, Barbara \| Krosky, Daniel Jason \| Querolle, Olivier Alexis Georges \| Patrick, Aaron Nathaniel \| Pilatte, Isabelle Noëlle Constance Patent Number: 10745409 (2020) Cite \| Source
6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors (patent) Wu, Tongfei \| Brehmer, Dirk \| Beke, Lijs \| Boeckx, An \| Diels, Gaston Stanislas Marcella \| Gilissen, Ronaldus Arnodus Hendrika Joseph \| Lawson, Edward Charles \| Pande, Vineet \| Paradé, Marcus Cornelis Bernardus Catharina \| Schepens, Wim Bert Griet \| ... \| Meerpoel, Lieven Patent Number: 10653711 (2020) Cited by (1) \| Cite \| Source
Fused bicyclic inhibitors of menin-MLL interaction (patent) Angibaud, Patrick Rene \| Pande, Vineet \| Herkert, Barbara \| Krosky, Daniel Jason \| Querolle, Olivier Alexis Georges \| Patrick, Aaron Nathaniel Patent Number: 10611778 (2020) Cite \| Source
Substituted thiohydantoin derivatives as androgen receptor antagonists (patent) Bignan, Gilles \| Connolly, Peter J. \| Hickson, Ian \| Meerpoel, Lieven \| Pande, Vineet \| Zhang, Zhuming \| Branch, Jonathan \| Rocaboy, Christian \| Trabalón Escolar, Luis B. Patent Number: 10501469 (2019) Cite \| Source
Preparation of 4′‐Spirocyclobutyl Nucleoside Analogues as Novel and Versatile Adenosine Scaffolds (journal article) Verhoeven, Jonas \| De Vleeschouwer, Freija \| Kong, Hanchu \| Van Hecke, Kristof \| Pande, Vineet \| Sun, Weimei \| Vos, Ann \| Wu, Tongfei \| Meerpoel, Lieven \| Thuring, Jan Willem \| Verniest, Guido Chemistry – A European Journal, volume 25, issue 67, pages 15419-15423 (2019). 10.1002/chem.201904574 Cited by (11) \| Cite \| Source
Design and synthesis of tetrahydropyridopyrimidine based Toll-Like Receptor (TLR) 7/8 dual agonists (journal article) McGowan, David C. \| Herschke, Florence \| Khamlichi, Mourad D. \| Rosauro, Mari Luz \| Benedicto, Sara M. Pérez \| Pauwels, Frederik \| Stoops, Bart \| Pande, Vineet \| Scholliers, Annick \| Van Schoubroeck, Bertrand \| ... \| Raboisson, Pierre Bioorganic & Medicinal Chemistry Letters, volume 28, issue 19, pages 3216-3221 (2018). 10.1016/j.bmcl.2018.08.015 Cited by (10) \| Cite \| Source
2,4-Diaminoquinazolines as Dual Toll-like Receptor (TLR) 7/8 Modulators for the Treatment of Hepatitis B Virus (journal article) Embrechts, Werner \| Herschke, Florence \| Pauwels, Frederik \| Stoops, Bart \| Last, Stefaan \| Pieters, Serge \| Pande, Vineet \| Pille, Geert \| Amssoms, Katie \| Smyej, Ilham \| ... \| McGowan, David Journal of Medicinal Chemistry, volume 61, issue 14, pages 6236-6246 (2018). 10.1021/acs.jmedchem.8b00643 Cited by (22) \| Cite \| Source
Substituted thiohydantoin derivatives as androgen receptor antagonists (patent) Bignan, Gilles \| Connolly, Peter J \| Hickson, Ian \| Meerpoel, Lieven \| Pande, Vineet \| Zhang, Zhuming \| Branch, Jonathan \| Rocaboy, Christian \| Trabalón Escolar, Luis B Patent Number: 10000502 (2018) Cite \| Source
Understanding the Complexity of Epigenetic Target Space (journal article) Pande, Vineet Journal of Medicinal Chemistry, volume 59, issue 4, pages 1299-1307 (2016). 10.1021/acs.jmedchem.5b01507 Cited by (28) \| Cite \| Source
Structural diversity of the epigenetics pocketome (journal article) Cabaye, Alexandre \| Nguyen, Kong T \| Liu, Lihua \| Pande, Vineet \| Schapira, Matthieu Proteins: Structure, Function, and Bioinformatics, volume 83, issue 7, pages 1316-1326 (2015). 10.1002/prot.24830 Cited by (9) \| Cite \| Source
Direct Covalent Modification as a Strategy to Inhibit Nuclear Factor-Kappa B (journal article) Pande, V. \| Sousa, S. \| Ramos, M. Current Medicinal Chemistry, volume 16, issue 32, pages 4261-4273 (2009). 10.2174/092986709789578222 Cited by (26) \| Cite \| Source
The Protein Kinase Inhibitor Balanol: Structure – Activity Relationships and Structure-Based Computational Studies (journal article) Pande, Vineet \| Ramos, Maria \| Gago, Federico Anti-Cancer Agents in Medicinal Chemistry, volume 8, issue 6, pages 638-645 (2008). 10.2174/187152008785133056 Cited by (23) \| Cite \| Source
Biological Evaluation, Chelation, and Molecular Modeling Studies of Novel Metal-Chelating Inhibitors of NF-κB-DNA Binding: Structure Activity Relationships (journal article) Sharma, Rakesh K. \| Chopra, Shilpa \| Sharma, Som D. \| Pande, Vineet \| Ramos, Maria J. \| Meguro, Kazuyuki \| Inoue, Jun-ichiro \| Otsuka, Masami Journal of Medicinal Chemistry, volume 49, issue 12, pages 3595-3601 (2006). 10.1021/jm050617x Cited by (16) \| Cite \| Source