Ajit Kandale

ScholarGPS® ID: 64408448725007

Affiliation
University of Queensland, Brisbane, Queensland, Australia, Australia
Affiliation History

Field
Physical Sciences and Mathematics
Discipline
Chemistry
Top Specialties
Medicinal Chemistry | Chemical Synthesis
Metrics Summary
Publication Count
19
Predicted Citations
418
Predicted h-index
13
Ranking

Publications and Citation History

Publications based on Top Specialties

Types of Publication

  • Publications
  • Books
  • Patents
  • NIH/NSF
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Analogues of the Herbicide, N -Hydroxy- N -isopropyloxamate, Inhibit Mycobacterium tuberculosis Ketol-Acid Reductoisomerase and Their Prodrugs Are Promising Anti-TB Drug Leads (journal article)
Kandale, Ajit | Patel, Khushboo | Hussein, Waleed M. | Wun, Shun Jie | Zheng, Shan | Tan, Lendl | West, Nicholas P. | Schenk, Gerhard | Guddat, Luke W. | McGeary, Ross P.
Journal of Medicinal Chemistry, volume 64, issue 3, pages 1670-1684 (2021).
10.1021/acs.jmedchem.0c01919
Cited by (12) | Cite | Source
Crystal Structures of Staphylococcus aureus Ketol‐Acid Reductoisomerase in Complex with Two Transition State Analogues that Have Biocidal Activity (journal article)
Patel, Khushboo M. | Teran, David | Zheng, Shan | Kandale, Ajit | Garcia, Mario | Lv, You | Schembri, Mark A. | McGeary, Ross P. | Schenk, Gerhard | Guddat, Luke W.
Chemistry – A European Journal, volume 23, issue 72, pages 18289-18295 (2017).
10.1002/chem.201704481
Cited by (22) | Cite | Source
Crystal structure of Mycobacterium tuberculosis ketol‐acid reductoisomerase at 1.0 Å resolution – a potential target for anti‐tuberculosis drug discovery (journal article)
Lv, You | Kandale, Ajit | Wun, Shun Jie | McGeary, Ross P. | Williams, Simon J. | Kobe, Bostjan | Sieber, Volker | Schembri, Mark A. | Schenk, Gerhard | Guddat, Luke W.
The FEBS Journal, volume 283, issue 7, pages 1184-1196 (2016).
10.1111/febs.13672
Cited by (30) | Cite | Source | Open Access
Synthesis & Biological Evaluation of 1, 3, 4- Oxadiazoles as Anticancer Agents (journal article)
D, Suryanarayana Raju | Kumar, T.N.V. Ganesh | Mathew, Jesil | Kandale, Ajit | Singla, Rajeev K
Indo Global Journal of Pharmaceutical Sciences, volume 05, issue 01, pages 01-05 (2015).
10.35652/IGJPS.2015.17
Cited by (4) | Cite | Source
Synthesis and in vitro cholesteryl ester transfer protein inhibitory activity of novel esters of 2, 10-dichloro-12H-dibenzo [d,g] 1,3-dioxocin-6-carboxylic acid (journal article)
Talluri, Sirishadevi | Kini, Suvarna G. | Kandale, Ajit | Kumar, Ganesh | Ohlyan, Renu
Medicinal Chemistry Research, volume 23, issue 10, pages 4491-4499 (2014).
10.1007/s00044-014-1021-1
Cited by (2) | Cite | Source
Pharmacophore modeling and 3D QSAR analysis of isothiazolidinedione derivatives as PTP1B inhibitors (journal article)
Deora, Girdhar Singh | Joshi, Prashant | Rathore, Vandana | Kumar, K. Lalith | Ohlyan, Renu | Kandale, Ajit
Medicinal Chemistry Research, volume 22, issue 7, pages 3478-3484 (2013).
10.1007/s00044-012-0349-7
Cited by (11) | Cite | Source
ChemInform Abstract: AgNO3 Mediated C—N Bond Forming Reaction: Synthesis of 3‐Substituted Benzothiazines as Potential COX Inhibitors. (journal article)
Rambabu, D. | Murthy, P. V. N. S. | Prasad, K. R. S. | Kandale, Ajit | Deora, Girdhar Singh | Rao, M. V. Basaveswara | Pal, Manojit
ChemInform, volume 44, issue 12 (2013).
10.1002/chin.201312167
Cite | Source
In vitro screening of dry fruit extracts of Piper attenuatum for antioxidant and anticancer activity (journal article)
Ohlyan, Renu | Kandale, Ajit | Deora, Girdhar Singh | Rathore, Vandana | Chahal, Jagbir
Medicinal Chemistry Research, volume 22, issue 3, pages 1365-1370 (2013).
10.1007/s00044-012-0122-y
Cited by (4) | Cite | Source
ChemInform Abstract: AlCl3 ‐Induced C—N Bond Formation Followed by Pd/C—Cu‐Mediated Coupling—Cyclization Strategy: Synthesis of Pyrrolo[2,3‐b]quinoxalines as Anticancer Agents. (journal article)
Prasad, Bagineni | Kumar, K. Shiva | Babu, P. Vijaya | Anusha, K. | Rambabu, D. | Kandale, Ajit | Vanaja, G. R. | Kalle, Arunasree M. | Pal, Manojit
ChemInform, volume 44, issue 8 (2013).
10.1002/chin.201308162
Cite | Source
Ultrasound-based approach to spiro-2,3-dihydroquinazolin-4(1H)-ones: their in vitro evaluation against chorismate mutase (journal article)
Rambabu, D. | Kiran Kumar, S. | Yogi Sreenivas, B. | Sandra, Sandhya | Kandale, Ajit | Misra, Parimal | Basaveswara Rao, M.V. | Pal, Manojit
Tetrahedron Letters, volume 54, issue 6, pages 495-501 (2013).
10.1016/j.tetlet.2012.11.057
Cited by (56) | Cite | Source
AlCl3 induced C–N bond formation followed by Pd/C–Cu mediated coupling–cyclization strategy: synthesis of pyrrolo[2,3-b]quinoxalines as anticancer agents (journal article)
Prasad, Bagineni | Shiva Kumar, K. | Vijaya Babu, P. | Anusha, K. | Rambabu, D. | Kandale, Ajit | Vanaja, G.R. | Kalle, Arunasree M. | Pal, Manojit
Tetrahedron Letters, volume 53, issue 45, pages 6059-6066 (2012).
10.1016/j.tetlet.2012.08.119
Cited by (27) | Cite | Source
AgNO3 mediated C–N bond forming reaction: synthesis of 3-substituted benzothiazines as potential COX inhibitors (journal article)
Rambabu, D. | Murthy, P.V.N.S. | Prasad, K.R.S. | Kandale, Ajit | Deora, Girdhar Singh | Basaveswara Rao, M.V. | Pal, Manojit
Tetrahedron Letters, volume 53, issue 48, pages 6577-6583 (2012).
10.1016/j.tetlet.2012.09.102
Cited by (18) | Cite | Source
Pd-mediated functionalization of polysubstituted pyrroles: Their evaluation as potential inhibitors of PDE4 (journal article)
Bhaskar Kumar, T. | Sumanth, Ch. | Vaishaly, S. | Srinivasa Rao, M. | Chandra Sekhar, K.B. | Meda, Chandana Lakshmi T. | Kandale, Ajit | Rambabu, D. | Rama Krishna, G. | Malla Reddy, C. | ... | Pal, Manojit
Bioorganic & Medicinal Chemistry Letters, volume 22, issue 17, pages 5639-5647 (2012).
10.1016/j.bmcl.2012.06.100
Cited by (18) | Cite | Source
C–N bond formation under Cu-catalysis: Synthesis and in vitro evaluation of N-aryl substituted thieno[2,3-d]pyrimidin-4(3H)-ones against chorismate mutase (journal article)
Adepu, Raju | Shiva Kumar, K. | Sandra, Sandhya | Rambabu, D. | Rama Krishna, G. | Malla Reddy, C. | Kandale, Ajit | Misra, Parimal | Pal, Manojit
Bioorganic & Medicinal Chemistry, volume 20, issue 17, pages 5127-5138 (2012).
10.1016/j.bmc.2012.07.011
Cited by (11) | Cite | Source
ChemInform Abstract: Design and Synthesis of 4‐Alkynyl Pyrazoles as Inhibitors of PDE4: A Practical Access via Pd/C—Cu Catalysis. (journal article)
Gorja, Dhilli Rao | Kumar, K. Shiva | Kandale, Ajit | Meda, Chandana Lakshmi T. | Parsa, Kishore V. L. | Mukkanti, K. | Pal, Manojit
ChemInform, volume 43, issue 34 (2012).
10.1002/chin.201234113
Cite | Source
Conformationally restricted novel pyrazole derivatives: Synthesis of 1,8-disubstituted 5,5-dimethyl-4,5-dihydro-1H-benzo[g]indazoles as a new class of PDE4 inhibitors (journal article)
Shyamsunder Reddy, T. | Shiva Kumar, K. | Meda, Chandana L.T. | Kandale, Ajit | Rambabu, D. | Rama Krishna, G. | Hariprasad, C. | Venugopala Rao, V. | Venkataiah, S. | Malla Reddy, C. | ... | Pal, Manojit
Bioorganic & Medicinal Chemistry Letters, volume 22, issue 9, pages 3248-3255 (2012).
10.1016/j.bmcl.2012.03.029
Cited by (10) | Cite | Source
Design and synthesis of 4-alkynyl pyrazoles as inhibitors of PDE4: A practical access via Pd/C–Cu catalysis (journal article)
Gorja, Dhilli Rao | Shiva Kumar, K. | Kandale, Ajit | Meda, Chandana Lakshmi T. | Parsa, Kishore V.L. | Mukkanti, K. | Pal, Manojit
Bioorganic & Medicinal Chemistry Letters, volume 22, issue 7, pages 2480-2487 (2012).
10.1016/j.bmcl.2012.02.008
Cited by (16) | Cite | Source
Novel thieno[2,3-d]pyrimidines: their design, synthesis, crystal structure analysis and pharmacological evaluation (journal article)
Adepu, Raju | Rambabu, D. | Prasad, Bagineni | Meda, Chandana Lakshmi T. | Kandale, Ajit | Rama Krishna, G. | Malla Reddy, C. | Chennuru, Lakshmi N. | Parsa, Kishore V. L. | Pal, Manojit
Organic & Biomolecular Chemistry, volume 10, issue 29, pages 5554- (2012).
10.1039/c2ob25420d
Cited by (28) | Cite | Source
Yb(OTf)3 mediated MCR: a new and regioselective approach towards polysubstituted pyrroles of pharmacological interest (journal article)
Reddy, G. Rajeshwar | Reddy, T. Ram | Joseph, Suju C. | Reddy, K. Sateesh | Meda, Chandana Lakshmi T. | Kandale, Ajit | Rambabu, D. | Krishna, G. Rama | Reddy, C. Malla | Parsa, Kishore V. L. | ... | Pal, Manojit
RSC Advances, volume 2, issue 24, pages 9142- (2012).
10.1039/c2ra21343e
Cited by (26) | Cite | Source