Peter J. Connolly | Scholar Profiles and Rankings

Publications and Citation History

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Gut-Restricted Selective Cyclooxygenase-2 (COX-2) Inhibitors for Chemoprevention of Colorectal Cancer (journal article) Zhang, Zhuming \| Ghosh, Avijit \| Connolly, Peter J. \| King, Peter \| Wilde, Thomas \| Wang, Jianyao \| Dong, Yawei \| Li, Xueliang \| Liao, Daohong \| Chen, Hao \| ... \| Evans, David C. Journal of Medicinal Chemistry, volume 64, issue 15, pages 11570-11596 (2021). 10.1021/acs.jmedchem.1c00890 Cited by (12) \| Cite \| Source
Spirocyclic Thiohydantoin Antagonists of F877L and Wild-Type Androgen Receptor for Castration-Resistant Prostate Cancer (journal article) Zhang, Zhuming \| Connolly, Peter J. \| Trabalón Escolar, Luis \| Rocaboy, Christian \| Pande, Vineet \| Meerpoel, Lieven \| Lim, Heng-Keang \| Branch, Jonathan R. \| Ondrus, Janine \| Hickson, Ian \| ... \| Bignan, Gilles ACS Medicinal Chemistry Letters, volume 12, issue 8, pages 1245-1252 (2021). 10.1021/acsmedchemlett.1c00032 Cited by (3) \| Cite \| Source
Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC) (journal article) Zhang, Zhuming \| Connolly, Peter J. \| Lim, Heng Keang \| Pande, Vineet \| Meerpoel, Lieven \| Teleha, Christopher \| Branch, Jonathan R. \| Ondrus, Janine \| Hickson, Ian \| Bush, Tammy \| ... \| Bignan, Gilles Journal of Medicinal Chemistry, volume 64, issue 2, pages 909-924 (2021). 10.1021/acs.jmedchem.0c01563 Cited by (17) \| Cite \| Source
The discovery of azetidine-piperazine di-amides as potent, selective and reversible monoacylglycerol lipase (MAGL) inhibitors (journal article) Zhu, Bin \| Connolly, Peter J. \| Zhang, Yue-Mei \| McDonnell, Mark E. \| Bian, Haiyan \| Lin, Shu-Chen \| Liu, Li \| Zhang, Sui-Po \| Chevalier, Kristen M. \| Brandt, Michael R. \| ... \| Macielag, Mark J. Bioorganic & Medicinal Chemistry Letters, volume 30, issue 14, pages 127243- (2020). 10.1016/j.bmcl.2020.127243 Cited by (12) \| Cite \| Source
The discovery of diazetidinyl diamides as potent and reversible inhibitors of monoacylglycerol lipase (MAGL) (journal article) Zhu, Bin \| Connolly, Peter J. \| Zhang, Sui-Po \| Chevalier, Kristen M. \| Milligan, Cynthia M. \| Flores, Christopher M. \| Macielag, Mark J. Bioorganic & Medicinal Chemistry Letters, volume 30, issue 12, pages 127198- (2020). 10.1016/j.bmcl.2020.127198 Cited by (7) \| Cite \| Source
Pharmacologic Characterization of JNJ-42226314, [1-(4-Fluorophenyl)indol-5-yl]-[3-[4-(thiazole-2-carbonyl)piperazin-1-yl]azetidin-1-yl]methanone, a Reversible, Selective, and Potent Monoacylglycerol Lipase Inhibitor (journal article) Wyatt, Ryan M. \| Fraser, Ian \| Welty, Natalie \| Lord, Brian \| Wennerholm, Michelle \| Sutton, Steven \| Ameriks, Michael K. \| Dugovic, Christine \| Yun, Sujin \| White, Allison \| ... \| Bonaventure, Pascal Journal of Pharmacology and Experimental Therapeutics, volume 372, issue 3, pages 339-353 (2020). 10.1124/jpet.119.262139 Cited by (15) \| Cite \| Source
Substituted thiohydantoin derivatives as androgen receptor antagonists (patent) Bignan, Gilles \| Connolly, Peter J. \| Hickson, Ian \| Meerpoel, Lieven \| Pande, Vineet \| Zhang, Zhuming \| Branch, Jonathan \| Rocaboy, Christian \| Trabalón Escolar, Luis B. Patent Number: 10501469 (2019) Cite \| Source
Discovery and optimization of a series of small-molecule allosteric inhibitors of MALT1 protease (journal article) Lu, Tianbao \| Connolly, Peter J. \| Philippar, Ulrike \| Sun, Weimei \| Cummings, Maxwell D. \| Barbay, Kent \| Gys, Luc \| Van Nuffel, Luc \| Austin, Nigel \| Bekkers, Mariette \| ... \| Edwards, James Bioorganic & Medicinal Chemistry Letters, volume 29, issue 23, pages 126743- (2019). 10.1016/j.bmcl.2019.126743 Cited by (10) \| Cite \| Source
Imidazolin-5-one derivative useful as FASN inhibitors for the treatment of cancer (patent) Connolly, Peter J \| Lu, Tianbao Patent Number: 10413545 (2019) Cited by (1) \| Cite \| Source
Imidazolin-5-one derivative useful as FASN inhibitors for the treatment of cancer (patent) Connolly, Peter J. \| Bignan, Gilles C. \| Lu, Tianbao \| Parker, Michael H. \| Ludovici, Donald W. \| Meyer, Christophe \| Meerpoel, Lieven \| Smans, Karine \| Rocaboy, Christian Patent Number: 10077261 (2018) Cite \| Source
Design and synthesis of a series of bioavailable fatty acid synthase (FASN) KR domain inhibitors for cancer therapy (journal article) Lu, Tianbao \| Schubert, Carsten \| Cummings, Maxwell D. \| Bignan, Gilles \| Connolly, Peter J. \| Smans, Karine \| Ludovici, Donald \| Parker, Michael H. \| Meyer, Christophe \| Rocaboy, Christian \| ... \| Meerpoel, Lieven Bioorganic & Medicinal Chemistry Letters, volume 28, issue 12, pages 2159-2164 (2018). 10.1016/j.bmcl.2018.05.014 Cited by (27) \| Cite \| Source
Substituted thiohydantoin derivatives as androgen receptor antagonists (patent) Bignan, Gilles \| Connolly, Peter J \| Hickson, Ian \| Meerpoel, Lieven \| Pande, Vineet \| Zhang, Zhuming \| Branch, Jonathan \| Rocaboy, Christian \| Trabalón Escolar, Luis B Patent Number: 10000502 (2018) Cite \| Source
Imidazolin-5-one derivative useful as FASN inhibitors for the treatment of cancer (patent) Connolly, Peter J \| Lu, Tianbao Patent Number: 9718813 (2017) Cited by (1) \| Cite \| Source
Benzamide derivative useful as FASN inhibitors for the treatment of cancer (patent) Connolly, Peter J \| Lu, Tianbao Patent Number: 9562035 (2017) Cite \| Source
Tetrahydroindazole derivatives as potent and peripherally selective cannabinoid-1 (CB1) receptor inverse agonists (journal article) Matthews, Jay M. \| McNally, James J. \| Connolly, Peter J. \| Xia, Mingde \| Zhu, Bin \| Black, Shawn \| Chen, Cailin \| Hou, Cuifen \| Liang, Yin \| Tang, Yuting \| Macielag, Mark J. Bioorganic & Medicinal Chemistry Letters, volume 26, issue 21, pages 5346-5349 (2016). 10.1016/j.bmcl.2016.09.025 Cited by (18) \| Cite \| Source
From Nanodiscs to Isotropic Bicelles: A Procedure for Solution Nuclear Magnetic Resonance Studies of Detergent-Sensitive Integral Membrane Proteins (journal article) Laguerre, Aisha \| Löhr, Frank \| Henrich, Erik \| Hoffmann, Beate \| Abdul-Manan, Norzehan \| Connolly, Peter J. \| Perozo, Eduardo \| Moore, Jonathan M. \| Bernhard, Frank \| Dötsch, Volker Structure, volume 24, issue 10, pages 1830-1841 (2016). 10.1016/j.str.2016.07.017 Cited by (27) \| Cite \| Source \| Open Access
Azetidinyl diamides as monoacylglycerol lipase inhibitors (patent) Bian, Haiyan \| Chevalier, Kristen \| Clemente, Jose \| Connolly, Peter J \| Flores, Christopher \| Lin, Shu-Chen \| Liu, Li \| Mabus, John \| Macielag, Mark \| McDonnell, Mark M \| ... \| Zhu, Bin Patent Number: 8962607 (2015) Cited by (6) \| Cite \| Source
A selective small molecule NOP (ORL-1 receptor) partial agonist for the treatment of anxiety (journal article) Ross, Tina Morgan \| Battista, Kathleen \| Bignan, Gilles C. \| Brenneman, Doug E. \| Connolly, Peter J. \| Liu, Jingchun \| Middleton, Steven A. \| Orsini, Michael \| Reitz, Allen B. \| Rosenthal, Dan I. \| ... \| Vaidya, Anil H. Bioorganic & Medicinal Chemistry Letters, volume 25, issue 3, pages 602-606 (2015). 10.1016/j.bmcl.2014.12.015 Cited by (14) \| Cite \| Source
Time-shared experiments for efficient assignment of triple-selectively labeled proteins (journal article) Löhr, Frank \| Laguerre, Aisha \| Bock, Christoph \| Reckel, Sina \| Connolly, Peter J. \| Abdul-Manan, Norzehan \| Tumulka, Franz \| Abele, Rupert \| Moore, Jonathan M. \| Dötsch, Volker Journal of Magnetic Resonance, volume 248 (2014). 10.1016/j.jmr.2014.09.014 Cited by (13) \| Cite \| Source \| Open Access
4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators (patent) Coats, Steven J. \| Bian, Haiyan \| Cai, Chaozhong \| DeCorte, Bart L. \| Liu, Li \| Macielag, Mark J. \| Dax, Scott L. \| Pitis, Philip M. \| Connolly, Peter J. \| He, Wei Patent Number: 8846655 (2014) Cited by (4) \| Cite \| Source