Christopher A. Teleha

ScholarGPS® ID: 35637736492790

Affiliation

Johnson & Johnson, New Brunswick, New Jersey, United States

Affiliation History

Field

Physical Sciences and Mathematics

Discipline

Chemistry

Top Specialties

Metrics Summary

Publication Count

Predicted Citations

1,948

Predicted h-index

Ranking

Publications and Citation History

Publications based on Top Specialties

Types of Publication

Publications
Books
Patents
NIH/NSF

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Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC) (journal article) Zhang, Zhuming \| Connolly, Peter J. \| Lim, Heng Keang \| Pande, Vineet \| Meerpoel, Lieven \| Teleha, Christopher \| Branch, Jonathan R. \| Ondrus, Janine \| Hickson, Ian \| Bush, Tammy \| ... \| Bignan, Gilles Journal of Medicinal Chemistry, volume 64, issue 2, pages 909-924 (2021). 10.1021/acs.jmedchem.0c01563 Cited by (17) \| Cite \| Source
Practical Synthesis of Ethyl 3-Fluoro-1-pyrrole-2-carboxylate: A Key Fragment of a Potent Drug Candidate against Hepatitis B Virus (journal article) René, Adeline \| Quilan, Maxime \| Deng, Yicheng \| Cheng, Yang \| Teleha, Christopher A. \| Raboisson, Pierre \| Bonfanti, Jean-François \| Fortin, Jérôme \| Charette, André. B. \| Pannecoucke, Xavier \| ... \| Jubault, Philippe Organic Process Research & Development, volume 24, issue 5, pages 792-801 (2020). 10.1021/acs.oprd.9b00382 Cited by (11) \| Cite \| Source
6-Benzhydryl-4-amino-quinolin-2-ones as Potent Cannabinoid Type 1 (CB1 ) Receptor Inverse Agonists and Chemical Modifications for Peripheral Selectivity (journal article) Zhang, Yue-Mei \| Greco, Michael N. \| Macielag, Mark J. \| Teleha, Christopher A. \| DesJarlais, Renee L. \| Tang, Yuting \| Ho, George \| Hou, Cuifen \| Chen, Cailin \| Zhao, Shuyuan \| ... \| Leonard, James Journal of Medicinal Chemistry, volume 61, issue 22, pages 10276-10298 (2018). 10.1021/acs.jmedchem.8b01467 Cited by (13) \| Cite \| Source
Crystals and process of making 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid (patent) Anzalone, Luigi \| Villani, Frank J. \| Teleha, Christopher A. \| Feibush, Penina \| Fegely, Barry Patent Number: 9789125 (2017) Cited by (1) \| Cite \| Source
Quinoline derivatives useful as CB-1 inverse agonists (patent) DeCorte, Bart \| Macielag, Mark \| Greco, Michael \| Zhang, Yue-Mei \| Teleha, Christopher Patent Number: 9464055 (2016) Cited by (2) \| Cite \| Source
Sulfonamides as TRPM8 modulators (patent) Branum, Shawn T \| Colburn, Raymond W \| Dax, Scott L \| Flores, Christopher M \| Jetter, Michele C \| Liu, Yi \| Ludovici, Donald \| Macielag, Mark J \| Matthews, Jay M \| McNally, James J \| ... \| Youngman, Mark A Patent Number: 9434711 (2016) Cite \| Source
Crystals and process of making 5-({[2-amino-3-(4-Carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid (patent) Anzalone, Luigi \| Villani, Frank J. \| Teleha, Christopher A. \| Feibush, Penina \| Fegely, Barry Patent Number: 9364489 (2016) Cited by (4) \| Cite \| Source
Process for the preparation of heterocyclic ester derivatives (patent) Bongartz, Jean-Pierre André Marc \| Stappers, Alfred Elisabeth \| Teleha, Christopher A. \| Weerts, Koen Johan Herman \| Wilson, Kenneth J. Patent Number: 9303046 (2016) Cite \| Source
Quinoline derivatives useful as CB-1 inverse agonists (patent) DeCorte, Bart \| Macielag, Mark \| Greco, Michael \| Zhang, Yue-Mei \| Teleha, Christopher Patent Number: 9266835 (2016) Cited by (3) \| Cite \| Source
Synthesis of Mavatrep: A Potent Antagonist of Transient Receptor Potential Vanilloid-1 (journal article) Wells, Kenneth M. \| Mehrman, Steven J. \| Abdel-Magid, Ahmed F. \| Ferraro, Caterina \| Scott, Lorraine \| Zhong, Hua Marlon \| Teleha, Christopher A. \| Ballentine, Scott \| Li, Xun \| Russell, Ronald K. \| ... \| Beauchamp, Derek A. Organic Process Research & Development, volume 19, issue 11, pages 1774-1783 (2015). 10.1021/acs.oprd.5b00271 Cited by (6) \| Cite \| Source
Process for the preparation of compounds useful as inhibitors of SGLT (patent) Filliers, Walter Ferdinand Maria \| Broeckx, Rudy Laurent Maria \| Nieste, Patrick Hubert J. \| Hatsuda, Masanori \| Yoshinaga, Masahiko \| Yada, Mitsuhiro \| Teleha, Christopher Patent Number: 9056850 (2015) Cite \| Source
Process for the preparation of C-FMS kinase inhibitors (patent) Kolodziejczyk, Krzysztof \| Stappers, Alfred Elisabeth \| Teleha, Christopher A. \| Weerts, Koen Johan Herman Patent Number: 9029352 (2015) Cite \| Source
Lab-Scale Preparation of a Novel Carbocyclic Chemokine Receptor Antagonist (journal article) Teleha, Christopher A. \| Branum, Shawn \| Zhang, Yongzheng \| Reuman, Michael E. \| Van Der Steen, Luc \| Verbeek, Marc \| Fawzy, Nagy \| Leo, Gregory C. \| Kang, Fu-An \| Cai, Chaozhong \| ... \| Vanbaelen, Hilde Organic Process Research & Development, volume 18, issue 12, pages 1622-1629 (2014). 10.1021/op500265z Cited by (7) \| Cite \| Source
Lab-Scale Preparation of a Novel Cyclopenta[b]furan Chemokine Receptor Antagonist (journal article) Teleha, Christopher A. \| Branum, Shawn \| Zhang, Yongzheng \| Reuman, Michael E. \| Van Der Steen, Luc \| Verbeek, Marc \| Fawzy, Nagy \| Leo, Gregory C. \| Winters, Michael P. \| Kang, Fu-An \| ... \| Vanbaelen, Hilde Organic Process Research & Development, volume 18, issue 12, pages 1630-1640 (2014). 10.1021/op500266w Cited by (8) \| Cite \| Source
Crystals and process of making 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid (patent) Anzalone, Luigi \| Villani, Frank J. \| Teleha, Christopher A. \| Feibush, Penina \| Fegely, Barry Patent Number: 8859604 (2014) Cited by (5) \| Cite \| Source
ChemInform Abstract: Synthesis of Substituted 2,4,5,6‐Tetrahydrocyclopenta[c]pyrazoles and 2,4,5,6‐Tetrahydropyrrolo[3,4‐c]pyrazoles by Intramolecular Nitrilimine Cycloaddition. (journal article) Winters, Michael P. \| Teleha, Christopher A. \| Sui, Zhihua ChemInform, volume 45, issue 35 (2014). 10.1002/chin.201435140 Cite \| Source
Sulfonamides as TRPM8 modulators (patent) Branum, Shawn T. \| Colburn, Raymond W. \| Dax, Scott L. \| Flores, Christopher M. \| Jetter, Michele C. \| Liu, Yi \| Ludovici, Donald \| Macielag, Mark J. \| Matthews, Jay M. \| McNally, James J. \| ... \| Youngman, Mark A. Patent Number: 8809327 (2014) Cited by (13) \| Cite \| Source
The discovery and SAR of cyclopenta[b]furans as inhibitors of CCR2 (journal article) Winters, Michael P. \| Teleha, Christopher A. \| Kang, Fu-An \| McComsey, David \| O’Neill, John C. \| Hou, Cuifen \| Kirchner, Thomas \| Wang, Ping \| Johnson, Dana \| Sui, Zhihua Bioorganic & Medicinal Chemistry Letters, volume 24, issue 9, pages 2137-2140 (2014). 10.1016/j.bmcl.2014.03.036 Cited by (5) \| Cite \| Source
Crystals and process of making 5-({(2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(-4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid (patent) Anzalone, Luigi \| Villani, Frank J. \| Teleha, Christopher A. \| Feibush, Penina \| Fegely, Barry Patent Number: 8691860 (2014) Cited by (6) \| Cite \| Source
Enantioselective process for preparing a substituted alkanoic acid (patent) Kinney, William A. \| Teleha, Christopher A. \| Ghosh, Shyamali \| Maryanoff, Bruce E. \| Grasa, Gabriela \| Zanotti-Gerosa, Antonio \| Medlock, Jonathan Alan Patent Number: 8680278 (2014) Cite \| Source