Shawn Branum

ScholarGPS® ID: 35211550788953

Affiliation

Janssen Pharmaceutica

Affiliation History

Field

Physical Sciences and Mathematics

Discipline

Chemistry

Top Specialties

Receptor Modulator | Medicinal Chemistry | Receptor Antagonist

Metrics Summary

Publication Count

Predicted Citations

385

Predicted h-index

Ranking

Publications and Citation History

Publications based on Top Specialties

Types of Publication

Publications
Books
Patents
NIH/NSF

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Substituted aza-bicyclic imidazole derivatives useful TRPM8 receptor modulators (patent) Player, Mark R. \| Calvo, Raul \| Chen, Jinsheng \| Meegalla, Sanath \| Parks, Daniel J. \| Parsons, William J. \| Ballentine, Scott \| Branum, Shawn Patent Number: 9718820 (2017) Cite \| Source
Process for the preparation of compounds useful as inhibitors of SGLT-2 (patent) Wells, Kenneth M. \| Russell, Ronald K. \| Li, Xun \| Branum, Shawn \| Beauchamp, Derek A. \| Nomura, Sumihiro \| Matsumura, Yosuke Patent Number: 9522931 (2016) Cite \| Source
Sulfonamides as TRPM8 modulators (patent) Branum, Shawn T \| Colburn, Raymond W \| Dax, Scott L \| Flores, Christopher M \| Jetter, Michele C \| Liu, Yi \| Ludovici, Donald \| Macielag, Mark J \| Matthews, Jay M \| McNally, James J \| ... \| Youngman, Mark A Patent Number: 9434711 (2016) Cite \| Source
Substituted aza-bicyclic imidazole derivatives useful as TRPM8 receptor modulators (patent) Player, Mark R. \| Calvo, Raul \| Chen, Jinsheng \| Meegalla, Sanath \| Parks, Daniel J. \| Parsons, William J. \| Ballentine, Scott \| Branum, Shawn Patent Number: 9409915 (2016) Cite \| Source
Substituted AZA-bicyclic imidazole derivatives useful as TRPM8 receptor modulators (patent) Player, Mark R \| Calvo, Raul \| Chen, Jinsheng \| Meegalla, Sanath \| Parks, Daniel J. \| Parsons, William J \| Ballentine, Scott \| Branum, Shawn Patent Number: 9023846 (2015) Cite \| Source
Lab-Scale Preparation of a Novel Carbocyclic Chemokine Receptor Antagonist (journal article) Teleha, Christopher A. \| Branum, Shawn \| Zhang, Yongzheng \| Reuman, Michael E. \| Van Der Steen, Luc \| Verbeek, Marc \| Fawzy, Nagy \| Leo, Gregory C. \| Kang, Fu-An \| Cai, Chaozhong \| ... \| Vanbaelen, Hilde Organic Process Research & Development, volume 18, issue 12, pages 1622-1629 (2014). 10.1021/op500265z Cited by (7) \| Cite \| Source
Lab-Scale Preparation of a Novel Cyclopenta[b]furan Chemokine Receptor Antagonist (journal article) Teleha, Christopher A. \| Branum, Shawn \| Zhang, Yongzheng \| Reuman, Michael E. \| Van Der Steen, Luc \| Verbeek, Marc \| Fawzy, Nagy \| Leo, Gregory C. \| Winters, Michael P. \| Kang, Fu-An \| ... \| Vanbaelen, Hilde Organic Process Research & Development, volume 18, issue 12, pages 1630-1640 (2014). 10.1021/op500266w Cited by (8) \| Cite \| Source
Sulfonamides as TRPM8 modulators (patent) Branum, Shawn T. \| Colburn, Raymond W. \| Dax, Scott L. \| Flores, Christopher M. \| Jetter, Michele C. \| Liu, Yi \| Ludovici, Donald \| Macielag, Mark J. \| Matthews, Jay M. \| McNally, James J. \| ... \| Youngman, Mark A. Patent Number: 8809327 (2014) Cited by (13) \| Cite \| Source
Substituted aza-bicyclic imidazole derivatives useful as TRPM8 receptor modulators (patent) Player, Mark R. \| Calvo, Raul \| Chen, Jinsheng \| Meegalla, Sanath \| Parks, Daniel \| Parsons, William \| Ballentine, Scott \| Branum, Shawn Patent Number: 8680098 (2014) Cited by (1) \| Cite \| Source
Process Development for Scale-Up of a Novel 3,5-Substituted Thiazolidine-2,4-dione Compound as a Potent Inhibitor for Estrogen-Related Receptor 1 (journal article) Li, Xun \| Russell, Ronald K. \| Spink, Jan \| Ballentine, Scott \| Teleha, Christopher \| Branum, Shawn \| Wells, Kenneth \| Beauchamp, Derek \| Patch, Raymond \| Huang, Hui \| ... \| Murray, William Organic Process Research & Development, volume 18, issue 2, pages 321-330 (2014). 10.1021/op400325r Cited by (14) \| Cite \| Source
FUSED CYCLOPENTYL ANTAGONISTS OF CCR2 (patent) Winters, Michael P. \| Branum, Shawn \| Fawzy, Nagy \| Kang, Fu-An \| Reuman, Michael \| Russell, Ronald K. \| Sui, Zhihua \| Teleha, Christopher A. Patent Number: 9150532 (2013) Cite \| Source
An Efficient Synthesis of 3-Substituted N -Glycoside Indoles Useful as Sodium-Dependent Glucose Transporter Inhibitors (journal article) Li, Xun \| Wells, Kenneth M. \| Branum, Shawn \| Damon, Sandra \| Youells, Scott \| Beauchamp, Derek A. \| Palmer, David \| Stefanick, Stephen \| Russell, Ronald K. \| Murray, William Organic Process Research & Development, volume 16, issue 11, pages 1727-1732 (2012). 10.1021/op3001355 Cited by (9) \| Cite \| Source
Sulfonamides as TRPM8 modulators (patent) Branum, Shawn T. \| Colburn, Raymond W. \| Dax, Scott L. \| Flores, Christopher M. \| Jetter, Michele C. \| Liu, Yi \| Ludovici, Donald \| Macielag, Mark J. \| Matthews, Jay M. \| McNally, James J. \| ... \| Youngman, Mark A. Patent Number: 8153682 (2012) Cited by (24) \| Cite \| Source
Design and Characterization of Optimized Adenosine A2A /A1 Receptor Antagonists for the Treatment of Parkinson's Disease (journal article) Shook, Brian C. \| Rassnick, Stefanie \| Wallace, Nathaniel \| Crooke, Jeffrey \| Ault, Mark \| Chakravarty, Devraj \| Barbay, J. Kent \| Wang, Aihua \| Powell, Mark T. \| Leonard, Kristi \| ... \| Jackson, Paul F. Journal of Medicinal Chemistry, volume 55, issue 3, pages 1402-1417 (2012). 10.1021/jm201640m Cited by (50) \| Cite \| Source
In Vivo Characterization of a Dual Adenosine A2A /A1 Receptor Antagonist in Animal Models of Parkinson’s Disease (journal article) Shook, Brian C. \| Rassnick, Stefanie \| Osborne, Melville C. \| Davis, Scott \| Westover, Lori \| Boulet, Jamie \| Hall, Daniel \| Rupert, Kenneth C. \| Heintzelman, Geoffrey R. \| Hansen, Kristin \| ... \| Jackson, Paul F. Journal of Medicinal Chemistry, volume 53, issue 22, pages 8104-8115 (2010). 10.1021/jm100971t Cited by (50) \| Cite \| Source
Optimization of arylindenopyrimidines as potent adenosine A2A/A1 antagonists (journal article) Shook, Brian C. \| Rassnick, Stefanie \| Chakravarty, Devraj \| Wallace, Nathaniel \| Ault, Mark \| Crooke, Jeffrey \| Barbay, J. Kent \| Wang, Aihua \| Leonard, Kristi \| Powell, Mark T. \| ... \| Jackson, Paul F. Bioorganic & Medicinal Chemistry Letters, volume 20, issue 9, pages 2868-2871 (2010). 10.1016/j.bmcl.2010.03.024 Cited by (12) \| Cite \| Source
Methylene amine substituted arylindenopyrimidines as potent adenosine A2A/A1 antagonists (journal article) Shook, Brian C. \| Rassnick, Stefanie \| Hall, Daniel \| Rupert, Kenneth C. \| Heintzelman, Geoffrey R. \| Hansen, Kristen \| Chakravarty, Devraj \| Bullington, James L. \| Scannevin, Robert H. \| Magliaro, Brian \| ... \| Jackson, Paul F. Bioorganic & Medicinal Chemistry Letters, volume 20, issue 9, pages 2864-2867 (2010). 10.1016/j.bmcl.2010.03.042 Cited by (24) \| Cite \| Source
Regio- and diastereoselective ring-opening of (S)-(−)-2-(trifluoromethyl)oxirane with chiral 2,5-disubstituted tetrahydroquinolines in hexafluoro-2-propanol (journal article) Li, Xun \| Russell, Ronald K. \| Chen, Hongfeng \| Zhang, Yongzheng \| Ballentine, Scott \| Spink, Jan \| Branum, Shawn \| Liu, Fuqiang \| Chen, Yanping \| Rammeloo, Thomas \| ... \| Murray, William V. Green Chemistry, volume 12, issue 9, pages 1548- (2010). 10.1039/c004726k Cited by (3) \| Cite \| Source
Synthesis of Tetracyclic Heterocompounds as Selective Estrogen Receptor Modulators. Part 2. Process Improvement for Scale-Up of 2,5,8-Substituted 11,12-Dihydro-5 H -6,13-dioxabenzo[3,4]cyclohepta-[1,2- a ]naphthalene Derivatives (journal article) Li, Xun \| Reuman, Michael \| Russell, Ronald K. \| Youells, Scott \| Beish, Sandra \| Hu, Zhiyong \| Branum, Shawn \| Jain, Nareshkumar \| Sui, Zhihua Organic Process Research & Development, volume 12, issue 1, pages 125-125 (2008). 10.1021/op700254f Cited by (3) \| Cite \| Source \| Open Access
Synthesis of Tetracyclic Heterocompounds as Selective Estrogen Receptor Modulators. Part 2. Process Improvement for Scale-Up Of 2,5,8-Substituted 11,12-Dihydro-5 H -6,13-dioxabenzo[3,4]cyclohepta-[1,2- a ]naphthalene Derivatives (journal article) Li, Xun \| Reuman, Michael \| Russell, Ronald K. \| Youells, Scott \| Beish, Sandra \| Hu, Zhiyong \| Branum, Shawn \| Jain, Nareshkumar \| Sui, Zhihua Organic Process Research & Development, volume 11, issue 4, pages 731-738 (2007). 10.1021/op700061x Cited by (8) \| Cite \| Source